9-amino-7-(substituted)-6-demethyl-6-deoxytetracyclines - Patent US5281628(A)

Filed: Oct 04, 1991

Published: Jan 25, 1994

Abstract

9-amino-7-(substituted amino)-6-demethyl-6-deoxytetracyclines having activity against a wide spectrum of organisms including organisms which are resistant to tetracyclines are disclosed. Also disclosed are intermediates and methods for making the novel compounds of the present invention.

Applicants

AMERICAN CYANAMID CO

Inventors

GLUZMAN YAKOV
HLAVKA JOSEPH J
LEE VING J
SUM PHAIK-ENG

Application Number

771697

Priority Claims

US77169791

Family Members

NO923856(D0) - NYE 9-AMINO-7-SUBSTITUERTE-6-DEMETYL-6-DEOKSYTETRACYKLINER

FI924453(D0) - NYA 9-AMINO-7-(SUBSTITUERAD)-6-DEMETYL-6-DEOXITETRACYKLINER

HU9203143(D0) - NEW 9-AMINO-7-(SUBSTITUTED)-6-DEMETHYL-6-DESOXI-TETRACYCLINES

IL103319(D0) - NOVEL 9-AMINO-7-(SUBSTITUTED)-6-DEMETHYL-6-DEOXYTETRACYCLINES

CA2079703(A1) - 9-AMINO-6-DEMETHYL-6-DESOXYTETRACYCLINES SUBSTITUEES EN 7

NO923856(A) - NYE 9-AMINO-7-SUBSTITUERTE-6-DEMETYL-6-DEOKSYTETRACYKLINER

FI924453(A) - NYA 9-AMINO-7-(SUBSTITUERAD)-6-DEMETYL-6-DEOXITETRACYKLINER

EP0535346(A1) - DesoxytÃ©tracycline-6, desmÃ©thyl-6, substituÃ©e 7, amino-9.

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US5281628(A) - 9-amino-7-(substituted)-6-demethyl-6-deoxytetracyclines

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Classification Codes

C07D333/36, C07C231/00, C07D213/74, C07D215/38, A61P31/04, C07D307/66, C07D215/00, C07D213/00, C07C231/12, C07D333/00, C07C237/00, C07C237/26, A61K31/47, A61K31/165, A61K31/65, A61P31/00, C07D307/00